MP-4222 | GRPR antagonist | Probechem Biochemicals

Chemical Structure : MP-4222

MP-4222 (MP4222)

Catalog No.: PC-27295Not For Human Use, Lab Use Only.

MP-4222 is a potent small molecule gastrin-releasing peptide receptor (GRPR) antagonist with binding IC50 of 21.2 nM, has equal selectivity over the neuromedin B receptor (NMBR).

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Biological Activity

MP-4222 is a potent small molecule gastrin-releasing peptide receptor (GRPR) antagonist with binding IC50 of 21.2 nM, has equal selectivity over the neuromedin B receptor (NMBR).

Physicochemical Properties

M.Wt	593.65
Formula	C32H34F3N5O3
Appearance	Solid
CAS No.
Storage	Solide Powder -20°C 12 Months; 4°C 6 Months	In Solvent -80°C 6 Months; -20°C 6 Months
Shipping
Solubility	10 mM in DMSO
Chemical Name/SMILES	(S)-N-((1-(2,6-difluoro-4-methoxyphenyl)cyclohexyl)methyl)-2-(3-(2-fluoropyridin-4-yl)ureido)-3-(1H-indol-3-yl)-2-methylpropanamide

References

1. Zhou M, et al. Med Chem Res. 2026 Jun;35(6):1119-1140.

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MP-4222 (MP4222)

Biological Activity

Physicochemical Properties

References

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