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Chemical Structure : Bantag-1 trifluoroacetate
Catalog No.: PC-61215Not For Human Use, Lab Use Only.
Bantag-1 trifluoroacetate is a potent, highly selective, peptide bombesin receptor subtype-3 (BRS-3) antagonist with IC50 of 2-8 nM for human and rodent BRS-3.
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Bantag-1 trifluoroacetate is a potent, highly selective, peptide bombesin receptor subtype-3 (BRS-3) antagonist with IC50 of 2-8 nM for human and rodent BRS-3.
Bantag-1 trifluoroacetate displays 1000-fold selectivity over hNMBR and hGRPR.
Bantag-1 trifluoroacetate increases food intake and produces an obesity phenotype in mice.
| M.Wt | ||
| Formula | C48H73N8O7 · xC2HF3O2 | |
| Appearance | Solid | |
| Storage |
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| Solubility |
10 mM in DMSO |
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1. Moreno P, et al. J Pharmacol Exp Ther. 2013 Oct;347(1):100-16.
2. Guan XM, et al. Cell Metab. 2010 Feb 3;11(2):101-12.
3. Feng Y, et al. Endocrinology. 2011 Nov;152(11):4106-15.
4. Nakamura T, et al. Biochem Pharmacol. 2016 Sep 1;115:64-76.
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