Chemical Structure : BX795
CAS No.:
702675-74-9
BX795
(BX 795, BX-795)
Catalog No. : PC-42629Not For Human Use, Lab Use Only.
BX795 is a potent and relatively specific PDK1 inhibitor with IC50 of 6 nM.
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Purity & Documentation Purity:
>98% (HPLC) Select Batch: PC-4262901
Biological Activity
BX795 is a potent and relatively specific PDK1 inhibitor with IC50 of 6 nM. TBK1 and IKKε with IC50 of 6 nM and 41 nM.
Physicochemical Properties
M.Wt
591.4677
Formula
C23H26IN7O2S
Appearance
Solid
CAS No.
Storage
Solide Powder
-20 °C 12 Months; 4°C 6 Months
In Solvent
-80 °C 6 Months; -20°C 6 Months
Shipping
Solubility
10 mM in DMSO
Chemical Name/SMILES
1-Pyrrolidinecarboxamide, N-[3-[[5-iodo-4-[[3-[(2-thienylcarbonyl)amino]propyl]amino]-2-pyrimidinyl]amino]phenyl]-
References
1. Clark K, et al. J Biol Chem.
2. Feldman RI, et al. J Biol Chem.
3. Frémond ML, et al. Arthritis Rheumatol.
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