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Request The Product List ofPDK1 PDK1

Cat. No. Product Name CAS No. Information
PC-62481

PS 210

1221962-86-2 PS 210 is a potent, specific activator of PDK1 that target the PIF-binding pocket of PDK1, does not alter the activity of any of the 121 kinases (S6K, PKB/Akt or GSK3)..
PC-60606

OSU-03013

742112-34-1 OSU-03013 (OSU 03013, OSU03013) is a novel potent, orally active 3-phosphoinositide-dependent kinase-1 (PDK-1) with IC50 of 2 uM.
PC-60605

OSU-03012

742112-33-0 OSU-03012 (AR-12) is a novel potent, orally active 3-phosphoinositide-dependent kinase-1 (PDK-1) with IC50 of 5 uM.
PC-42781

BX-912

702674-56-4 BX-912 (BX912) is a potent, selective and ATP-competitive inhibitor of PDK1 with IC50 of 26 nM.
PC-42629

BX795

702675-74-9 BX795 is a potent and relatively specific PDK1 inhibitor with IC50 of 6 nM.
PC-73258

PDK-1 agonist PS48

1180676-32-7 PDK-1 agonist PS48 is a small molecule allosteric PDK-1 agonist, PS48 is active at 10 nM to 1 μM in restoring normal insulin-dependent Akt activation and in mitigating Aβi peptide toxicity.
PC-63030

BX-320

702676-93-5 BX-320 is a potent, selective and ATP-competitive inhibitor of PDK1 with IC50 of 30 nM, >20-fold selectivity over PKA.

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