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Baclofen

Chemical Structure : Baclofen

CAS No.: 1134-47-0

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Baclofen

Catalog No.: PC-46124Not For Human Use, Lab Use Only.

Baclofen is a derivative of the neurotransmitter GABA that acts as a GABAB receptor agonist.

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2 g $88 In stock
5 g $138 In stock
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Purity & Documentation Purity: >98% (HPLC) Select Batch:

Biological Activity

Baclofen is a derivative of the neurotransmitter GABA that acts as a GABAB receptor agonist.
Baclofen also blocks α2δ subunit-containing voltage-dependent calcium channel (VDCC) with Ki of 156 uM.
Baclofen is a neurotransmitter inhibitor by blocking the release of excitatory transmitters.
Baclofen serves as a central nervous system depressant and skeletal muscle relaxant.

Physicochemical Properties

M.Wt 213.6608
Formula C10H12ClNO2
Appearance Solid
CAS No.
Storage
Solide Powder
-20 °C 12 Months; 4°C 6 Months
In Solvent
-80 °C 6 Months; -20°C 6 Months
Shipping
Solubility

DMSO: < 7.8 mg/mL
Chemical Name/SMILES

Benzenepropanoic acid, β-(aminomethyl)-4-chloro-

References

1. Zvejniece L, et al. Pharmacol Biochem Behav. 2015 Oct;137:23-9.

2. Carter LP, et al. Pharmacol Ther. 2009 Jan;121(1):100-14.

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