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Bergaptol

Chemical Structure : Bergaptol

CAS No.: 486-60-2

Bergaptol (5-Hydroxypsoralen, 4-Hydroxybergapten)

Catalog No.: PC-45969Not For Human Use, Lab Use Only.

Bergaptol is a natural furanocoumarin that is found to be a potent inhibitor of debenzylation activity of CYP3A4 enzyme with IC50 of 24.92 uM.

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Purity & Documentation Purity: >98% (HPLC) Select Batch:

Biological Activity

Bergaptol is a natural furanocoumarin that is found to be a potent inhibitor of debenzylation activity of CYP3A4 enzyme with IC50 of 24.92 uM.
Bergaptol shows very good radical scavenging activity.

Physicochemical Properties

M.Wt 202.1629
Formula C11H6O4
Appearance Solid
CAS No.
Storage
Solide Powder
-20 °C 12 Months; 4°C 6 Months
In Solvent
-80 °C 6 Months; -20°C 6 Months
Shipping
Solubility

DMSO: < 2.1 mg/mL

Chemical Name/SMILES

7H-Furo[3,2-g][1]benzopyran-7-one, 4-hydroxy-

References

1. Girennavar B, et al. Bioorg Med Chem. 2007 Jun 1;15(11):3684-91.

2. Messer A, et al. Food Chem Toxicol. 2012 Mar;50(3-4):756-60.

3. Uesawa Y, et al. Pharmazie. 2011 Jul;66(7):525-8.

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