Cat. No. |
Product Name |
Information |
PC-20618 |
Decursin
CYP2J2 inhibitor
|
Decursin ((+)-Decursin) is a potent anti-tumor agent and a potent protein kinase C activator, induces apoptosis and cell cycle arrest at G1 phase. |
PC-20617 |
LKY-047
CYP2J2 inhibitor
|
LKY-047 (LKY047) is a potent, highly selective and reversible competitive cytochrome P450 CYP2J2 (CYP2J2) inhibitor with IC50 of 1.7 uM. |
PC-49015 |
DLCI-1 dihydrochloride
CYP2A6 inhibitor
|
DLCI-1 dihydrochloride is a potent and selective CYP2A6 inhibitor with IC50 of 17 nM, 15-765-fold selectivity other major hepatic CYP enzymes. |
PC-49014 |
DLCI-1
CYP2A6 inhibitor
|
DLCI-1 is a potent and selective CYP2A6 inhibitor with IC50 of 17 nM, 15-765-fold selectivity other major hepatic CYP enzymes. |
PC-72852 |
VID400
CYP24A1 inhibitor
|
VID400 (NVP-VID400, SDZ285-428) is a potent, selective inhibitor of CYP24A1. |
PC-72686 |
DX308
CYP26 inhibitor
|
DX308 is a potent, selective dual CYP26A1/B1 inhibitor and retinoic acid metabolism blocking agent. |
PC-72684 |
DX314
CYP26B1 inhibitor
|
DX314 is a potent, specific CYP26B1 inhibitor with IC50 of 108 nM, >15-fold selectivity over CYP26A1. |
PC-72679 |
8-BOA
CYP4Z1 inhibitor
|
8-BOA is a selective and potent mechanism-based inactivator of breast cancer-associated CYP4Z1. |
PC-35319 |
HET0016
CYP4A inhibitor
|
HET0016 (HET-0016) is a potent, selective inhibitor of CYP4A, potently inhibits the formation of 20-HETE with IC50 of 8.9 nM in human renal microsomes. |
PC-42617 |
Cobicistat
CYP3A inhibitor
|
Cobicistat (GS-9350) is a pharmacoenhancer that acts as potent and selective inhibitor of human CYP3A with IC50 of 30-285 nM. |
PC-21449 |
Dual CYP19A1/CYP11B2 inhibitor X21
CYP19A1/CYP11B2 inhibitor
|
Dual CYP19A1/CYP11B2 inhibitor X21 is a potent and selective dual inhibitor of aromatase (CYP19A1) and aldosterone synthase (CYP11B2) with IC50 of 2.3 nM and 29 nM, respectively. |
PC-21418 |
TPP-IOA
Cyt c peroxidase inhibitor
|
TPP-IOA is a specific inhibitor of cytochrome c (cyt c) peroxidase activity, inhibits peroxidase activity of cardiolipin-induced cytochrome c peroxidase activity with IC50 of 5 uM. |