Bizine |CAS:1591932-50-1 Probechem Biochemicals

Chemical Structure : Bizine

Bizine

Catalog No.: PC-62871Not For Human Use, Lab Use Only.

Bizine is a phenelzine analog that inhibits LSD1 with Ki of 59 nM, displays 23-fold, 63-fold, and >100-fold selectivity for LSD-1 over MAOA, MAOB, and LSD2 respectively.

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Biological Activity

Bizine is a phenelzine analog that inhibits LSD1 with Ki of 59 nM, displays 23-fold, 63-fold, and >100-fold selectivity for LSD-1 over MAOA, MAOB, and LSD2 respectively.
Bizine induces bulk histone H3 lysine 4 dimethylation in LNCaP cancer cells (EC50=2 uM).
Bizine protects neurons exposed to oxidative stress at 0.5 uM.

Physicochemical Properties

M.Wt	297.402
Formula	C18H23N3O
Appearance	Solid
CAS No.
Storage	Solide Powder -20 °C 12 Months; 4°C 6 Months	In Solvent -80 °C 6 Months; -20°C 6 Months
Shipping
Solubility	10 mM in DMSO
Chemical Name/SMILES	N-[4-(2-hydrazinylethyl)phenyl]-benzenebutanamide

References

1. Prusevich P, et al. ACS Chem Biol. 2014 Jun 20;9(6):1284-93.

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Bizine

Biological Activity

Physicochemical Properties

References

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