CBP bromodomain inhibitor |CAS:2161356-61-0 Probechem Biochemicals

Chemical Structure : CBP bromodomain inhibitor 17

CBP bromodomain inhibitor 17 (CBP-IN-17)

Catalog No.: PC-63543Not For Human Use, Lab Use Only.

CBP-IN-17 is a potent, selective CBP bromodomain inhibitor with IC50 of 69 nM, displays exquisite selectivity over BRD4(1) (IC50=18 uM) and the broader bromodomain family.

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Biological Activity

CBP-IN-17 is a potent, selective CBP bromodomain inhibitor with IC50 of 69 nM, displays exquisite selectivity over BRD4(1) (IC50=18 uM) and the broader bromodomain family.

Physicochemical Properties

M.Wt	426.486
Formula	C22H20F2N4OS
Appearance	Solid
CAS No.
Storage	Solide Powder -20 °C 12 Months; 4°C 6 Months	In Solvent -80 °C 6 Months; -20°C 6 Months
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Solubility	10 mM in DMSO
Chemical Name/SMILES	5-(7-(difluoromethyl)-6-(1-methyl-1H-pyrazol-4-yl)-3,4-dihydroquinolin-1(2H)-yl)-3-methylbenzo[d]thiazol-2(3H)-one

References

1. Bronner SM, et al. J Med Chem. 2017 Dec 28;60(24):10151-10171.

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CBP bromodomain inhibitor 17 (CBP-IN-17)

Biological Activity

Physicochemical Properties

References

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