CBR-470-2

Chemical Structure : CBR-470-2

CAS No.: 2416095-00-4

Catalog No.: PC-24726Not For Human Use, Lab Use Only.

CBR-470-2 is a small molecule inhibitor of glycolytic enzyme phosphoglycerate kinase 1 (PGK1), activates NRF2 signaling in vitro and in vivo.

Packing	Price	Stock
2 mg	$198	In stock
5 mg	$348	In stock
10 mg	$548	In stock
25 mg		Get quote
100 mg		Get quote

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Biological Activity

CBR-470-2 is a small molecule inhibitor of glycolytic enzyme phosphoglycerate kinase 1 (PGK1), activates NRF2 signaling in vitro and in vivo.
CBR-470-2 attenuated NF-κB signaling, decreasing transcriptional output in response to several canonical NF-κB activating stimuli.

Physicochemical Properties

M.Wt	402.26
Formula	C12H13Cl2NO6S2
Appearance	Solid
CAS No.
Storage	Solide Powder -20°C 12 Months; 4°C 6 Months	In Solvent -80°C 6 Months; -20°C 6 Months
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Solubility	10 mM in DMSO
Chemical Name/SMILES	Glycine, N-[(3R,4S)-4-[(3,4-dichlorophenyl)sulfonyl]tetrahydro-1,1-dioxido-3-thienyl]-, rel-

References

1. Bollong MJ, et, al. Nature. 2018 Oct;562(7728):600-604.

2. Caroline Stanton, et al. bioRxiv [Preprint]. 2025 May 16:2025.05.13.653579.

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CBR-470-2

Biological Activity

Physicochemical Properties

References

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