CCG-232601 | MRTF/SRF inhibitor | Probechem Biochemicals

Chemical Structure : CCG-232601

CAS No.: 1922099-21-5

CCG-232601 (CCG232601)

Catalog No.: PC-62824Not For Human Use, Lab Use Only.

CCG-232601 is a potent (IC50=0.55 uM), orally bioavailable inhibitor of Rho/MRTF/SRF transcriptional pathway that target transcriptional factor MRTF.

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5 mg	$398	In stock
10 mg	$588	In stock
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Biological Activity

CCG-232601 is a potent (IC50=0.55 uM), orally bioavailable inhibitor of Rho/MRTF/SRF transcriptional pathway that target transcriptional factor MRTF.
CCG-232601 inhibits the development of bleomycin-induced dermal fibrosis in mice when administered at 50mg/kg.

Physicochemical Properties

M.Wt	455.89
Formula	C24H20ClF2N3O2
Appearance	Solid
CAS No.
Storage	Solide Powder -20 °C 12 Months; 4°C 6 Months	In Solvent -80 °C 6 Months; -20°C 6 Months
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Solubility	10 mM in DMSO
Chemical Name/SMILES	N-(4-chlorophenyl)-5,5-difluoro-1-(3-(pyridin-4-yl)benzoyl)piperidine-3-carboxamide

References

1. Hutchings KM, et al. Bioorg Med Chem Lett. 2017 Apr 15;27(8):1744-1749.

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CCG-232601 (CCG232601)

Biological Activity

Physicochemical Properties

References

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