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CCG-232601

Chemical Structure : CCG-232601

CAS No.: 1922099-21-5

CCG-232601 (CCG232601)

Catalog No.: PC-62824Not For Human Use, Lab Use Only.

CCG-232601 is a potent (IC50=0.55 uM), orally bioavailable inhibitor of Rho/MRTF/SRF transcriptional pathway that target transcriptional factor MRTF.

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Purity & Documentation Purity: >98% (HPLC) Select Batch:

Biological Activity

CCG-232601 is a potent (IC50=0.55 uM), orally bioavailable inhibitor of Rho/MRTF/SRF transcriptional pathway that target transcriptional factor MRTF.
CCG-232601 inhibits the development of bleomycin-induced dermal fibrosis in mice when administered at 50mg/kg.

Physicochemical Properties

M.Wt 455.89
Formula C24H20ClF2N3O2
Appearance Solid
CAS No.
Storage
Solide Powder
-20 °C 12 Months; 4°C 6 Months
In Solvent
-80 °C 6 Months; -20°C 6 Months
Shipping
Solubility

10 mM in DMSO

Chemical Name/SMILES

N-(4-chlorophenyl)-5,5-difluoro-1-(3-(pyridin-4-yl)benzoyl)piperidine-3-carboxamide

References

1. Hutchings KM, et al. Bioorg Med Chem Lett. 2017 Apr 15;27(8):1744-1749.

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