CCG257081 | MRTF/SRF inhibitor | Probechem Biochemicals

Chemical Structure : CCG257081

CCG257081 (CCG-257081)

Catalog No.: PC-23604Not For Human Use, Lab Use Only.

CCG-257081 is a small molecule MRTF/SRF pathway inhibitor, shows direct binding to pirin with ITC KD value of 8.6 uM, inhibits melanoma metastasis and bleomycin-induced fibrosis.

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Biological Activity

CCG-257081 is a small molecule MRTF/SRF pathway inhibitor, shows direct binding to pirin with ITC KD value of 8.6 uM, inhibits melanoma metastasis and bleomycin-induced fibrosis.

Physicochemical Properties

M.Wt	473.88
Formula	C24H19ClF3N3O2
Appearance	Solid
CAS No.
Storage	Solide Powder -20°C 12 Months; 4°C 6 Months	In Solvent -80°C 6 Months; -20°C 6 Months
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Solubility	10 mM in DMSO
Chemical Name/SMILES	N-(4-chlorophenyl)-5,5-difluoro-1-(3-fluoro-5-(pyridin-4-yl)benzoyl)piperidine-3-carboxamide

References

1. Erika M Lisabeth, et al. ACS Pharmacol Transl Sci. 2019 Apr 12;2(2):92-100.

2. Panesso-Gómez S, et al. bioRxiv [Preprint]. 2024 Nov 17:2024.11.15.623825.

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CCG257081 (CCG-257081)

Biological Activity

Physicochemical Properties

References

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