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CJ-1639

Chemical Structure : CJ-1639

CAS No.: 1313759-88-4

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CJ-1639 (CJ1639)

Catalog No.: PC-72157Not For Human Use, Lab Use Only.

CJ-1639 (CJ1639) is a potent, highly selective dopamine D3 receptor (D3R) full agonist with Ki of 0.5 nM, >5,000-fold selectivity over D1 and D2 receptors in binding assays.

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Purity & Documentation Purity: >98% (HPLC) Select Batch:

    Biological Activity

    CJ-1639 (CJ1639) is a potent, highly selective dopamine D3 receptor (D3R) full agonist with Ki of 0.5 nM, >5,000-fold selectivity over D1 and D2 receptors in binding assays.
    CJ-1639 binds to human D3 receptor with a K(i) value of 3.61 nM and displays over >1000-fold selectivity over human D1 and D2 receptors.
    CJ-1639 is an excellent pharmacological tool to elucidate the role of the D3 receptor in different neurological conditions in animal models.

    Physicochemical Properties

    M.Wt 478.655
    Formula C27H34N4O2S
    Appearance Solid
    CAS No.
    Storage
    Solide Powder
    -20°C 12 Months; 4°C 6 Months
    In Solvent
    -80°C 6 Months; -20°C 6 Months
    Shipping
    Solubility

    10 mM in DMSO
    Chemical Name/SMILES

    N-((1R,3r)-3-(2-(((S)-2-amino-4,5,6,7-tetrahydrobenzo[d]thiazol-6-yl)(propyl)amino)ethyl)-3-hydroxycyclobutyl)-2-naphthamide

    References

    1. Jianyong Chen, et al. ACS Med Chem Lett. 2011 Aug 11;2(8):620-625.

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