CPI-268456 |CAS:1380087-86-4 Probechem Biochemicals

Chemical Structure : CPI-268456

CAS No.: 1380087-86-4

Catalog No.: PC-70026Not For Human Use, Lab Use Only.

CPI-268456 is a small molecule ligand of bromodomain-containing protein 4 (BRD4), binds to BRD4 with IC50 of 0.5 uM in cell-free assays.

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Biological Activity

CPI-268456 is a small molecule ligand of bromodomain-containing protein 4 (BRD4), binds to BRD4 with IC50 of 0.5 uM in cell-free assays.

CPI-268456 inhibits LPS-induced IL-6 secretion in THP-1 cells with IC50 of 0.5 uM.

M.Wt	400.259
Formula	C20H15Cl2N3O2
Appearance	Solid
CAS No.
Storage	Solide Powder -20 °C 12 Months; 4°C 6 Months	In Solvent -80 °C 6 Months; -20°C 6 Months
Shipping
Solubility	10 mM in DMSO
Chemical Name/SMILES	(S)-2-(8-chloro-6-(4-chlorophenyl)-1-methyl-4H-benzo[c]isoxazolo[4,5-e]azepin-4-yl)acetamide

1. Albrecht, B.K., Audia, J.E., Côté, A., et al. Bromodomain inhibitors and uses thereof. (2012).