You are here:Home-Chemical Inhibitors & Agonists-Epigenetics-Bromodomain-CPI-268456
CPI-268456

Chemical Structure : CPI-268456

CAS No.: 1380087-86-4

CPI-268456 (CPI 268456, CPI268456)

Catalog No.: PC-70026Not For Human Use, Lab Use Only.

CPI-268456 is a small molecule ligand of bromodomain-containing protein 4 (BRD4), binds to BRD4 with IC50 of 0.5 uM in cell-free assays.

Packing Price Stock Quantity
5 mg $158 In stock
10 mg $248 In stock
25 mg Get quote
50 mg Get quote
100 mg Get quote

Bulk size, bulk discount!

E-mail: sales@probechem.com

Tech Support: tech@probechem.com

Purity & Documentation Purity: >98% (HPLC) Select Batch:

Biological Activity

CPI-268456 is a small molecule ligand of bromodomain-containing protein 4 (BRD4), binds to BRD4 with IC50 of 0.5 uM in cell-free assays.
CPI-268456 inhibits LPS-induced IL-6 secretion in THP-1 cells with IC50 of 0.5 uM.

Physicochemical Properties

M.Wt 400.259
Formula C20H15Cl2N3O2
Appearance Solid
CAS No.
Storage
Solide Powder
-20 °C 12 Months; 4°C 6 Months
In Solvent
-80 °C 6 Months; -20°C 6 Months
Shipping
Solubility

10 mM in DMSO

Chemical Name/SMILES

(S)-2-(8-chloro-6-(4-chlorophenyl)-1-methyl-4H-benzo[c]isoxazolo[4,5-e]azepin-4-yl)acetamide

References

1. Albrecht, B.K., Audia, J.E., Côté, A., et al. Bromodomain inhibitors and uses thereof. (2012).

Copyright © 2022 probechem.com. All Rights Reserved. probechem Copyright

Contact Us sales@probechem.com

Bulk Inquiry

* Indicates a Required FieldYour information is safe with us.

  • *Product name:
  • *Applicant name:
  • *Email address:
  • *Organization name:
  • *Requested quantity:
  • *Country:
  • *Additional Information:

Get Quote

* Indicates a Required FieldYour information is safe with us.

  • *Product name:
  • *Applicant name:
  • *Email address:
  • *Organization name:
  • *Requested quantity:
  • *Country:
  • Additional Information: