Chemical Structure : CPN-351
CAS No.: 3057171-63-5
Catalog No.: PC-26901Not For Human Use, Lab Use Only.
CPN-351 is a potent, selective pentapeptide antagonist of Neuromedin U Receptor 1 (NMUR1) with pA2 and KB values of 7.35 and 45 nM, respectively, selective over NMUR2 with 6.38 and 421 nM, respectively.
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|---|---|---|---|
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| 10 mg | $248 | In stock | |
| 25 mg | $428 | In stock | |
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CPN-351 is a potent, selective pentapeptide antagonist of Neuromedin U Receptor 1 (NMUR1) with pA2 and KB values of 7.35 and 45 nM, respectively, selective over NMUR2 with 6.38 and 421 nM, respectively.
| M.Wt | 912.13 | |
| Formula | C45H61N13O6S | |
| Appearance | Solid | |
| Storage |
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| Solubility |
10 mM in DMSO |
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| Chemical Name/SMILES |
(S)-1-(((S)-2-((S)-3-(1H-indol-3-yl)-2-(N-methyl-2-(thiophen-2-yl)acetamido)propanamido)-2-methyl-3-phenylpropanoyl)-L-arginyl)-N-((S)-1-amino-5-guanidino-1-oxopentan-2-yl)pyrrolidine-2-carboxamide |
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1. Kentaro Takayama, et al. ACS Med Chem Lett. 2024 May 24;15(6):885-891.

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