Catalog No.: PC-28128Not For Human Use, Lab Use Only.
CPUY192002 is a potent protein-protein interaction (PPI) inhibitor of Keap1-Nrf2 with KD of 3.59 nM, effectively disrupts the Nrf2-Keap1 interaction with an EC50 of 28.6 nM in FP assays, also activates the Nrf2 transcription activity in the cell-based ARE-luciferase reporter assay.
CPUY192002 is a potent protein-protein interaction (PPI) inhibitor of Keap1-Nrf2 with KD of 3.59 nM, effectively disrupts the Nrf2-Keap1 interaction with an EC50 of 28.6 nM in FP assays, also activates the Nrf2 transcription activity in the cell-based ARE-luciferase reporter assay.
