Chemical Structure : CX-6258
CAS No.:
1202916-90-2
CX-6258
(CX6258, CX 6258)
Catalog No. : PC-45415Not For Human Use, Lab Use Only.
CX-6258 (CX6258) is a potent, selective, and orally efficacious pan-Pim inhibitor with IC50 of 5/25/16 nM for Pim1/2/3, respectively.
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Purity & Documentation Purity:
>98% (HPLC) Select Batch: PC-4541501
Biological Activity
CX-6258 (CX6258) is a potent, selective, and orally efficacious pan-Pim inhibitor with IC50 of 5/25/16 nM for Pim1/2/3, respectively.
Physicochemical Properties
M.Wt
461.9401
Formula
C26H24ClN3O3
Appearance
Solid
CAS No.
Storage
Solide Powder
-20 °C 12 Months; 4°C 6 Months
In Solvent
-80 °C 6 Months; -20°C 6 Months
Shipping
Solubility
10 mM in DMSO
Chemical Name/SMILES
2H-Indol-2-one, 5-chloro-3-[[5-[3-[(hexahydro-4-methyl-1H-1,4-diazepin-1-yl)carbonyl]phenyl]-2-furanyl]methylene]-1,3-dihydro-, (3E)-
References
1. Haddach M, et al. ACS Med Chem Lett.
2. Padmanabhan A, et al. J Cell Biochem.
3. Rebello RJ, et al. Clin Cancer Res.
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