CXCR7 agonist 1

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Chemical Structure : CXCR7 agonist 1

Catalog No.: PC-38669Not For Human Use, Lab Use Only.

CXCR agonist 1 is a potent, selective, small molecule agonist of CXCR7 (ACKR3), induces β-arrestin recruitment to CXCR7 and Akt activation, inhibits CXCL12-induced tube formation in HUVECs with EC50 of 0.96 nM.

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Purity & Documentation Purity: >98% (HPLC) Select Batch:

Biological Activity

CXCR7 agonist 1 is a potent, selective, small molecule agonist of CXCR7 (ACKR3), induces β-arrestin recruitment to CXCR7 and Akt activation, inhibits CXCL12-induced tube formation in HUVECs with EC50 of 0.96 nM.

Physicochemical Properties

M.Wt	447.332
Formula	C24H19BrN2O2
Appearance	Solid
CAS No.
Storage	Solide Powder -20°C 12 Months; 4°C 6 Months	In Solvent -80°C 6 Months; -20°C 6 Months
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Solubility	10 mM in DMSO
Chemical Name/SMILES	1-((6-bromopyridin-2-yl)methyl)-3-(3,4-dimethylbenzoyl)quinolin-4(1H)-one

References

1. Ayako Uto-Konomi, et al. Biochem Biophys Res Commun. 2013 Feb 22;431(4):772-6.

2. Adlere I, et al. Mol Pharmacol. 2019 Dec;96(6):737-752.

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CXCR7 agonist 1

Biological Activity

Physicochemical Properties

References

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