CXCR7 agonist 1

You are here:Home-Chemical Inhibitors & Agonists-GPCR-Chemokine Receptor (CCR and CXCR)-CXCR7 agonist 1

Chemical Structure : CXCR7 agonist 1

Catalog No.: PC-38669Not For Human Use, Lab Use Only.

CXCR agonist 1 is a potent, selective, small molecule agonist of CXCR7 (ACKR3), induces β-arrestin recruitment to CXCR7 and Akt activation, inhibits CXCL12-induced tube formation in HUVECs with EC50 of 0.96 nM.

Packing	Price	Stock	Quantity
25 mg		Get quote
50 mg		Get quote
100 mg		Get quote

Get Quotation Now

* Please select Quantity before adding items.

or Bulk Inquiry

Bulk size, bulk discount!

E-mail: sales@probechem.com

Tech Support: tech@probechem.com

Purity & Documentation Purity: >98% (HPLC) Select Batch:

Biological Activity

CXCR7 agonist 1 is a potent, selective, small molecule agonist of CXCR7 (ACKR3), induces β-arrestin recruitment to CXCR7 and Akt activation, inhibits CXCL12-induced tube formation in HUVECs with EC50 of 0.96 nM.

Physicochemical Properties

M.Wt	447.332
Formula	C24H19BrN2O2
Appearance	Solid
CAS No.
Storage	Solide Powder -20°C 12 Months; 4°C 6 Months	In Solvent -80°C 6 Months; -20°C 6 Months
Shipping
Solubility	10 mM in DMSO
Chemical Name/SMILES	1-((6-bromopyridin-2-yl)methyl)-3-(3,4-dimethylbenzoyl)quinolin-4(1H)-one

References

1. Ayako Uto-Konomi, et al. Biochem Biophys Res Commun. 2013 Feb 22;431(4):772-6.

2. Adlere I, et al. Mol Pharmacol. 2019 Dec;96(6):737-752.

Overnight Delivery
Fast & Safe Delivery Worldwide
Rewards Program

About Us

Our Services

Site Map

Join with Us
Product Use Citations

Pharmacological Glossary Abbreviations

Abbreviations

Quality Manual

Inquiry Form
How to Order

Terms & Conditions

Credit Card Payment

Shipping Rates & Policies

Privacy Policy
sales@probechem.com

CXCR7 agonist 1

Biological Activity

Physicochemical Properties

References

Bulk Inquiry

* Indicates a Required FieldYour information is safe with us.

Get Quote

* Indicates a Required FieldYour information is safe with us.