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Cat. No. Product Name CAS No. Information
PC-73030

CCR4-IN-31

2206788-99-8 CCR4-IN-31 (CCR4-351) is a potent, selective, orally bioavailable CCR4 antagonist with IC50 of 40 nM (Ca2+ flux).
PC-35600

LIT-927

2172879-52-4 LIT-927 (LIT927) is the first selective, locally and orally active CXCL12 neutraligand with Ki of 267 nM for CXCL12-TR binding inhibition.
PC-35572

CCR6 inhibitor 35

2437547-04-9 CCR6 inhibitor 35 is a potent and selective CCR6 inhibitor with IC50 of 6.0 nM (hCCR6).
PC-35514

AZ084

929300-19-6 AZ084 (AZ-084) is a potent, selective, allosteric, orally available CCR8 antagonist with Ki of 0.9 nM.
PC-63440

R243

688352-84-3 R243 is a potent, small molecule CCR8 antagonist that inhibits CCR8 signaling and chemotaxis, inhibits CCL1-induced Ca2+ flux and CCL1-driven peritoneal macrophages aggregation at 0.2 uM.
PC-62989

Elubrixin

688763-64-6 Elubrixin (SB-656933, GSK-656933) is a potent, selective, competitive and reversible CXCR2 antagonist.
PC-62762

AZD-4818

1003566-93-5 AZD-4818 is a highly potent, selective CCR1 antagonist with pIC50 of 8.6, inhibits chemotaxia of human monocytes to MIP-1α in a concentration-dependent manner.

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