Chemical Structure : Calhex231 hydrochloride
CAS No.:
2387505-78-2
Calhex231 hydrochloride
(Calhex-231 hydrochloride)
Catalog No. : PC-25683Not For Human Use, Lab Use Only.
Calhex231 hydrochloride is a potent negative allosteric modulator / antagonist of CaSR that blocks calcium-mediated activation with IC50 of 0.39 uM.
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Purity & Documentation Purity:
>98% (HPLC) Select Batch: PC-2568301
Biological Activity
Calhex231 hydrochloride is a potent negative allosteric modulator / antagonist of CaSR that blocks calcium-mediated activation with IC50 of 0.39 uM.
Physicochemical Properties
M.Wt
443.41
Formula
C25H28Cl2N2O
Appearance
Solid
CAS No.
Storage
Solide Powder
-20°C 12 Months; 4°C 6 Months
In Solvent
-80°C 6 Months; -20°C 6 Months
Shipping
Solubility
10 mM in DMSO
Chemical Name/SMILES
4-Chloro-N-((1S,2S)-2-(((R)-1-(naphthalen-1-yl)ethyl)amino)cyclohexyl)benzamide hydrochloride
References
1. Petrel C, et al. J Biol Chem. 2003 Dec 5;278(49):49487-94.
2. Weston AH, et al. Circ Res. 2005 Aug 19;97(4):391-8.
3. Kessler A, et al. J Med Chem. 2006 Aug 24;49(17):5119-28.
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