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Cat. No. Product Name CAS No. Information
PC-35260

GSK3004774

2138814-32-9 GSK3004774 (GSK-3004774) is a potent, nonabsorbable, gastrointestinally-restricted agonist agonist of calcium-sensing receptor (CaSR) with pEC50 of 7.3.
PC-63560

Velcalcetide

1262780-97-1 Velcalcetide (AMG-416, Velcalcetide, Etelcalcetide, KAI-4169) is a potent, peptide agonist of CaSR, dose-dependenty increases IP1 accumulation with EC50 of 25 uM in cell based assays.
PC-62910

Calindol hydrochloride

729610-18-8 Calindol hydrochloride is a calcimimetic acting agent and positive allosteric modulator (agonist) of CaSR with EC50 of 0.31 uM (stimulated 3H IP accumulation in CHO cells at 2 mM Ca2+).
PC-62909

Tecalcet

148717-54-8 Tecalcet (R-568.
PC-62908

Tecalcet hydrochloride

177172-49-5 Tecalcet (R-568.
PC-62907

AC-265347

1253901-26-6 AC-265347 is a calcimimetic acting agent and highly efficacious, orally active allosteric agonist (PAM) of CaSR with IC50 of 10 nM in PI hydrolysis assays.
PC-62905

Calhex-231

652973-93-8 Calhex-231 is a potent negative allosteric modulator of CaSR that blocks calcium-mediated activation with IC50 of 0.39 uM.

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