| Cat. No. |
Product Name |
CAS No. |
Information |
| PC-35260 |
GSK3004774
|
2138814-32-9 |
GSK3004774 (GSK-3004774) is a potent, nonabsorbable, gastrointestinally-restricted agonist agonist of calcium-sensing receptor (CaSR) with pEC50 of 7.3. |
| PC-63560 |
Velcalcetide
|
1262780-97-1 |
Velcalcetide (AMG-416, Velcalcetide, Etelcalcetide, KAI-4169) is a potent, peptide agonist of CaSR, dose-dependenty increases IP1 accumulation with EC50 of 25 uM in cell based assays. |
| PC-62910 |
Calindol hydrochloride
|
729610-18-8 |
Calindol hydrochloride is a calcimimetic acting agent and positive allosteric modulator (agonist) of CaSR with EC50 of 0.31 uM (stimulated 3H IP accumulation in CHO cells at 2 mM Ca2+). |
| PC-62909 |
Tecalcet
|
148717-54-8 |
Tecalcet (R-568. |
| PC-62908 |
Tecalcet hydrochloride
|
177172-49-5 |
Tecalcet (R-568. |
| PC-62907 |
AC-265347
|
1253901-26-6 |
AC-265347 is a calcimimetic acting agent and highly efficacious, orally active allosteric agonist (PAM) of CaSR with IC50 of 10 nM in PI hydrolysis assays. |
| PC-62905 |
Calhex-231
|
652973-93-8 |
Calhex-231 is a potent negative allosteric modulator of CaSR that blocks calcium-mediated activation with IC50 of 0.39 uM. |
