| Cat. No. |
Product Name |
Information |
| PC-42415 |
NPS-2143 hydrochloride
CaSR antagonist
|
NPS-2143 (SB262470A) hydrochloride is a potent, selective and orally active CaSR antagonist with IC50 of 43 nM. |
| PC-42051 |
NPS-2143
CaSR antagonist
|
NPS-2143 (SB262470) is a potent, selective and orally active CaSR antagonist with IC50 of 43 nM. |
| PC-45942 |
Cinacalcet hydrochloride
CaSR activator
|
Cinacalcet (AMG 073) hydrochloride is a calcimimetic agent that acts as an allosteric activator of CaSR. |
| PC-45941 |
Cinacalcet
CaSR agonist
|
Cinacalcet (AMG073) is a calcimimetic agent that acts as an allosteric activator of CaSR with EC50 of 51 nM. |
| PC-62910 |
Calindol hydrochloride
|
Calindol hydrochloride is a calcimimetic acting agent and positive allosteric modulator (agonist) of CaSR with EC50 of 0.31 uM (stimulated 3H IP accumulation in CHO cells at 2 mM Ca2+). |
| PC-45220 |
Strontium ranelate
|
A strontium(II) salt of ranelic acid that stimulates CaSR and leads to the differentiation of pre-osteoblast to osteoblast, increases the bone formation. |
| PC-45852 |
CaSR-IN-10a
|
A potent CaSR antagonist with IC50 of 4.4 nM in CaSR FLIPR assay.. |
