Calcium-sensing Receptor (CaSR) (inhibitors, antagonists, agonists)-ProbeChem.com

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Cat. No.	Product Name	Information
PC-42415	NPS-2143 hydrochloride CaSR antagonist	NPS-2143 (SB262470A) hydrochloride is a potent, selective and orally active CaSR antagonist with IC50 of 43 nM.
PC-42051	NPS-2143 CaSR antagonist	NPS-2143 (SB262470) is a potent, selective and orally active CaSR antagonist with IC50 of 43 nM.
PC-45942	Cinacalcet hydrochloride CaSR activator	Cinacalcet (AMG 073) hydrochloride is a calcimimetic agent that acts as an allosteric activator of CaSR.
PC-45941	Cinacalcet CaSR agonist	Cinacalcet (AMG073) is a calcimimetic agent that acts as an allosteric activator of CaSR with EC50 of 51 nM.
PC-62910	Calindol hydrochloride	Calindol hydrochloride is a calcimimetic acting agent and positive allosteric modulator (agonist) of CaSR with EC50 of 0.31 uM (stimulated 3H IP accumulation in CHO cells at 2 mM Ca2+).
PC-45220	Strontium ranelate	A strontium(II) salt of ranelic acid that stimulates CaSR and leads to the differentiation of pre-osteoblast to osteoblast, increases the bone formation.
PC-45852	CaSR-IN-10a	A potent CaSR antagonist with IC50 of 4.4 nM in CaSR FLIPR assay..

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