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Cenacitinib

Chemical Structure : Cenacitinib

CAS No.: 2641636-52-2

Cenacitinib (VTX-958, VTX958)

Catalog No.: PC-24937Not For Human Use, Lab Use Only.

Cenacitinib (VTX 958) is a potent, highly selective, allosteric and orally bioavailable inhibitor of tyrosine kinase 2 (TYK2).

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Purity & Documentation Purity: >98% (HPLC)

Biological Activity

Cenacitinib (VTX 958) is a potent, highly selective, allosteric and orally bioavailable inhibitor of tyrosine kinase 2 (TYK2).

Physicochemical Properties

M.Wt 431.40
Formula C19H19F2N7O3
Appearance Solid
CAS No.
Storage
Solide Powder
-20°C 12 Months; 4°C 6 Months
In Solvent
-80°C 6 Months; -20°C 6 Months
Shipping
Solubility

10 mM in DMSO

Chemical Name/SMILES

1-(5-((7-fluoro-2,3-dihydrobenzo[b][1,4]dioxin-5-yl)amino)-7-(methylamino)pyrazolo[1,5-a]pyrimidin-3-yl)-3-((1R,2S)-2-fluorocyclopropyl)urea

References

1. Patent WO2024151992 A1.

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