Cenobamate | GABAA PAM | Probechem Biochemicals

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Chemical Structure : Cenobamate

Cenobamate (YKP-3089, YKP3089)

Catalog No.: PC-28240Not For Human Use, Lab Use Only.

Cenobamate (YKP3089) is an antiepileptic compound that acts as a positive allosteric modulator of high-affinity GABAA receptors, potentiates GABA-induced currents (IGABA) in acutely isolated CA3 pyramidal cells with EC50 of 164 uM.

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Purity & Documentation Purity: >98% (HPLC)

Biological Activity

Physicochemical Properties

M.Wt	267.67
Formula	C10H10ClN5O2
Appearance	Solid
CAS No.
Storage	Solide Powder -20°C 12 Months; 4°C 6 Months	In Solvent -80°C 6 Months; -20°C 6 Months
Shipping
Solubility	10 mM in DMSO
Chemical Name/SMILES	[(1R)-1-(2-chlorophenyl)-2-(tetrazol-2-yl)ethyl] carbamate

References

1. Sperling MR, et al. Epilepsia. 2020 Jun;61(6):1099-1108.

2. Sharma R, et al. Eur J Pharmacol. 2020 Jul 15;879:173117.

3. Nakamura M, et al. Eur J Pharmacol. 2019 Jul 15;855:175-182.

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Cenobamate (YKP-3089, YKP3089)

Biological Activity

Physicochemical Properties

References

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