Chemical Structure : Cobicistat
CAS No.:
1004316-88-4
Cobicistat
(GS-9350, GS9350)
Catalog No. : PC-42617Not For Human Use, Lab Use Only.
Cobicistat (GS-9350) is a pharmacoenhancer that acts as potent and selective inhibitor of human CYP3A with IC50 of 30-285 nM.
Packing Price Stock Quantity 5 mg $88 In stock 0 1 2 3 4 5 10 mg $138 In stock 0 1 2 3 4 5 25 mg $228 In stock 0 1 2 3 4 5 50 mg $378 In stock 0 1 2 3 4 5 100 mg Get quote 0 1 2 3 4 5
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Purity & Documentation Purity:
>98% (HPLC) Select Batch: PC-4261701
Biological Activity
Cobicistat (GS-9350) is a pharmacoenhancer that acts as potent and selective inhibitor of human CYP3A with IC50 of 30-285 nM.
Physicochemical Properties
M.Wt
776.0227
Formula
C40H53N7O5S2
Appearance
Solid
CAS No.
Storage
Solide Powder
-20 °C 12 Months; 4°C 6 Months
In Solvent
-80 °C 6 Months; -20°C 6 Months
Shipping
Solubility
DMSO: ≥ 29 mg/mL
Chemical Name/SMILES
2,7,10,12-Tetraazatridecanoic acid, 12-methyl-13-[2-(1-methylethyl)-4-thiazolyl]-9-[2-(4-morpholinyl)ethyl]-8,11-dioxo-3,6-bis(phenylmethyl)-, 5-thiazolylmethyl ester, (3R,6R,9S)-
References
1. Xu L, et al. ACS Med Chem Lett.
2. Lepist EI, et al. Antimicrob Agents Chemother.
3. Stray KM, et al. Antimicrob Agents Chemother.
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