Chemical Structure : DASA-58
CAS No.:
1203494-49-8
DASA-58
(DASA58, DASA 58)
Catalog No. : PC-45611Not For Human Use, Lab Use Only.
A potent activator of PKM2 (pyruvate kinase M2) with AC50 of 38 nM.
Packing Price Stock Quantity 5 mg $88 In stock 0 1 2 3 4 5 10 mg $128 In stock 0 1 2 3 4 5 25 mg $218 In stock 0 1 2 3 4 5 50 mg $358 In stock 0 1 2 3 4 5 100 mg Get quote 0 1 2 3 4 5
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Purity & Documentation Purity:
>98% (HPLC) Select Batch: PC-4561101
Biological Activity
DASA-58 is a potent activator of PKM2 (pyruvate kinase M2) with AC50 of 38 nM; shows no activity on PKM1 in vitro.
Physicochemical Properties
M.Wt
453.5324
Formula
C19H23N3O6S2
Appearance
Solid
CAS No.
Storage
Solide Powder
-20 °C 12 Months; 4°C 6 Months
In Solvent
-80 °C 6 Months; -20°C 6 Months
Shipping
Solubility
DMSO: ≥ 35 mg/mL
Chemical Name/SMILES
Benzenamine, 3-[[4-[(2,3-dihydro-1,4-benzodioxin-6-yl)sulfonyl]hexahydro-1H-1,4-diazepin-1-yl]sulfonyl]-
References
1. Anastasiou D, et al. Nat Chem Biol
2. Palsson-McDermott EM, et al. Cell Metab
3. Giannoni E, et al. Oncotarget
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