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DC591053

Chemical Structure : DC591053

CAS No.: 3017184-78-7

DC591053 (DC 591053)

Catalog No.: PC-20022Not For Human Use, Lab Use Only.

DC591053 (DC 591053) is a selective small molecule agonist of relaxin family peptide receptor 4 (RXFP4) with pEC50  of 7.24  and pKi  of  6.95, shows no activity against RXFP3.

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    Biological Activity

    DC591053 (DC 591053) is a selective small molecule agonist of relaxin family peptide receptor 4 (RXFP4) with pEC50  of 7.24  and pKi  of  6.95, shows no activity against RXFP3.

    Physicochemical Properties

    M.Wt 493.60
    Formula C28H35N3O5
    Appearance Solid
    CAS No.
    Storage
    Solide Powder
    -20°C 12 Months; 4°C 6 Months
    In Solvent
    -80°C 6 Months; -20°C 6 Months
    Shipping
    Solubility

    10 mM in DMSO

    Chemical Name/SMILES

    (S)-(7-ethoxy-6-methoxy-1-(2-(5-methoxy-1H-indol-3-yl)ethyl)-3,4-dihydroisoquinolin-2(1H)-yl)(morpholino)methanone

    References

    1. Yan Chen, et al. Nat Commun. 2023 Jan 30;14(1):492.

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