Welcome to ProbeChem!Global Supplier of Chemical Probes, Inhibitors & Agonists.
Chemical Structure : DDP-38003 dihydrochloride
CAS No.: 1831167-98-6
Catalog No.: PC-45657Not For Human Use, Lab Use Only.
DDP-38003 dihydrochloride is a potent, selective and orally available inhibitor of histone lysine-specific demethylase 1A (KDM1A/LSD1) with IC50 of 84 nM.
| Packing | Price | Stock | Quantity |
|---|---|---|---|
| 5 mg | $158 | In stock | |
| 10 mg | $248 | In stock | |
| 25 mg | $398 | In stock | |
| 50 mg | Get quote | ||
| 100 mg | Get quote |
Bulk size, bulk discount!
E-mail: sales@probechem.com
Tech Support: tech@probechem.com
DDP-38003 dihydrochloride is a potent, selective and orally available inhibitor of histone lysine-specific demethylase 1A (KDM1A/LSD1) with IC50 of 84 nM.
DDP-38003 weakly inhibits MAO-A and has no activity for KDM1B and MAO-B (IC50>30 uM).
DDP-38003 is orally bioactive and exhibits in vivo efficacy in mouse leukemia model.
| M.Wt | 423.37922 | |
| Formula | C21H28Cl2N4O | |
| Appearance | Solid | |
| Storage |
|
|
| Solubility |
DMSO: ≥ 29 mg/mL |
|
| Chemical Name/SMILES |
Benzamide, N-[4-[(1S,2R)-2-aminocyclopropyl]phenyl]-4-(4-methyl-1-piperazinyl)-, hydrochloride (1:2) |
|
1. Vianello P, et al. J Med Chem. 2016 Feb 25;59(4):1501-17.
Copyright © 2022 probechem.com. All Rights Reserved. probechem Copyright
