DNA-PK inhibitor 78

Chemical Structure : DNA-PK inhibitor 78

Catalog No.: PC-22698Not For Human Use, Lab Use Only.

DNA-PK inhibitor 78 is a potent, selective DNA-PK inhibitor with IC50 of 7.95 nM, >200-fold selective over PI3Kα and >800-fold over other PI3Ks and mTOR.

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Biological Activity

DNA-PK inhibitor 78 is a potent, selective DNA-PK inhibitor with IC50 of 7.95 nM, >200-fold selective over PI3Kα and >800-fold over other PI3Ks and mTOR.

Physicochemical Properties

M.Wt	368.44
Formula	C20H24N4O3
Appearance	Solid
CAS No.
Storage	Solide Powder -20°C 12 Months; 4°C 6 Months	In Solvent -80°C 6 Months; -20°C 6 Months
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Solubility	10 mM in DMSO
Chemical Name/SMILES	6-((4-Methoxy-2-methylphenyl)amino)-3-methyl-1-(tetrahydro-2H-pyran-4-yl)-1,3-dihydro-2H-imidazo[4,5-c]pyridin-2-one

References

1. Hong CR, et al. J Med Chem. 2024 Jul 15. doi: 10.1021/acs.jmedchem.4c01120.

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