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DNA-PK inhibitor 78

Chemical Structure : DNA-PK inhibitor 78

CAS No.: 2766001-96-9

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DNA-PK inhibitor 78

Catalog No.: PC-22698Not For Human Use, Lab Use Only.

DNA-PK inhibitor 78 is a potent, selective DNA-PK inhibitor with IC50 of 7.95 nM, >200-fold selective over PI3Kα and >800-fold over other PI3Ks and mTOR.

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Purity & Documentation Purity: >98% (HPLC)

Biological Activity

DNA-PK inhibitor 78 is a potent, selective DNA-PK inhibitor with IC50 of 7.95 nM, >200-fold selective over PI3Kα and >800-fold over other PI3Ks and mTOR.

Physicochemical Properties

M.Wt 368.44
Formula C20H24N4O3
Appearance Solid
CAS No.
Storage
Solide Powder
-20°C 12 Months; 4°C 6 Months
In Solvent
-80°C 6 Months; -20°C 6 Months
Shipping
Solubility

10 mM in DMSO
Chemical Name/SMILES

6-((4-Methoxy-2-methylphenyl)amino)-3-methyl-1-(tetrahydro-2H-pyran-4-yl)-1,3-dihydro-2H-imidazo[4,5-c]pyridin-2-one

References

1. Hong CR, et al. J Med Chem. 2024 Jul 15. doi: 10.1021/acs.jmedchem.4c01120.

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