DPTN dihydrochloride | A3AR antagonist

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Chemical Structure : DPTN dihydrochloride

CAS No.: 325767-87-1

DPTN dihydrochloride (MRS7799)

Catalog No.: PC-28427Not For Human Use, Lab Use Only.

DPTN dihydrochloride (MRS7799) is a potent and selective A3 adenosine receptor (A3AR) antagonist with of 1.65, 9.61, and 8.53 nM for human, mouse, and rat A3AR respectively, and EC50 of 63.8 nM in A3AR-βarr2 recruitment assay.

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10 mg	$148	In stock
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Purity & Documentation Purity: >98% (HPLC) Select Batch:

Biological Activity

Physicochemical Properties

M.Wt	459.39
Formula	C22H20Cl2N4OS
Appearance	Solid
CAS No.
Storage	Solide Powder -20°C 12 Months; 4°C 6 Months	In Solvent -80°C 6 Months; -20°C 6 Months
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Solubility	10 mM in DMSO
Chemical Name/SMILES	N-(4-(3,5-Dimethylphenyl)-5-(pyridin-4-yl)thiazol-2-yl)nicotinamide dihydrochloride

References

1. Zhan-Guo Gao, et al. Purinergic Signal. 2021 Dec;17(4):737-746.

2. Suresh RR, et al. ACS Med Chem Lett. 2022 Mar 2;13(4):623-631.

3. Pottie E, et al. ACS Pharmacol Transl Sci. 2023 Aug 9;6(9):1266-1274.

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DPTN dihydrochloride (MRS7799)

Biological Activity

Physicochemical Properties

References

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