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DS-6930

Chemical Structure : DS-6930

CAS No.: 1242328-82-0

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DS-6930 (DS 6930;DS6930)

Catalog No.: PC-35674Not For Human Use, Lab Use Only.

DS-6930 (DS 6930, DS6930) is a novel potent, selective PPARγ agonist with EC50 of 41 nM, Emax-68%.

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Purity & Documentation Purity: >98% (HPLC) Select Batch:

    Biological Activity

    DS-6930 (DS 6930, DS6930) is a novel potent, selective PPARγ agonist with EC50 of 41 nM, Emax-68%.
    DS-6930 significantly recruits several cofactors, such as RIP140 and PGC1, in cofactor recruitment assays.
    DS-6930 demonstrates high PPARγ agonist potency with robust plasma glucose reduction, maintains diminished PPARγ-related adverse effects upon toxicological evaluation in vivo, and demonstrated no hepatotoxicity.

    Physicochemical Properties

    M.Wt 403.438
    Formula C23H21N3O4
    Appearance Solid
    CAS No.
    Storage
    Solide Powder
    -20 °C 12 Months; 4°C 6 Months
    In Solvent
    -80 °C 6 Months; -20°C 6 Months
    Shipping
    Solubility

    10 mM in DMSO
    Chemical Name/SMILES

    3-((6-((3,5-dimethylpyridin-2-yl)oxy)-1-methyl-1H-benzo[d]imidazol-2-yl)methoxy)benzoic acid calcium salt

    References

    1. Shinozuka T, et al. Bioorg Med Chem. 2018 Oct 1;26(18):5099-5117.

    2. Shinozuka T, et al. Bioorg Med Chem. 2018 Oct 1;26(18):5079-5098.

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