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DS69910557

Chemical Structure : DS69910557

CAS No.: 3032750-17-4

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DS69910557 (DS 69910557)

Catalog No.: PC-38658Not For Human Use, Lab Use Only.

DS69910557 is a highly potent, selective orally available human parathyroid hormone receptor 1 (hPTHR1) antagonist with IC50 of 0.08 uM.

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Purity & Documentation Purity: >98% (HPLC) Select Batch:

    Biological Activity

    DS69910557 is a highly potent, selective orally available human parathyroid hormone receptor 1 (hPTHR1) antagonist with IC50 of 0.08 uM.
    DS69910557 demonstrated in vivo potency to decrease the plasma calcium concentration in rats upon oral administration.

    Physicochemical Properties

    M.Wt 611.539
    Formula C32H33Cl2FN4O3
    Appearance Solid
    CAS No.
    Storage
    Solide Powder
    -20°C 12 Months; 4°C 6 Months
    In Solvent
    -80°C 6 Months; -20°C 6 Months
    Shipping
    Solubility

    10 mM in DMSO
    Chemical Name/SMILES

    (1r,4r)-4-(((1-(4-(2,9-dichloro-5,5-dimethyl-6-oxo-5,6-dihydro-7H-benzo[b]pyrido[3,2-d]azepin-7-yl)phenyl)-3-fluoroazetidin-3-yl)methyl)amino)cyclohexane-1-carboxylic acid

    References

    1. Yoshikazu Arai, et al. Bioorg Med Chem. 2022 Jun 15;64:116763.

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