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DS96432529

Chemical Structure : DS96432529

CAS No.: 868067-30-5

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DS96432529 (DS 96432529)

Catalog No.: PC-72664Not For Human Use, Lab Use Only.

DS96432529 (DS 96432529) is a potent and orally active bone anabolic agent with EC200 value of 0.024 ug/mL.

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Purity & Documentation Purity: >98% (HPLC) Select Batch:

    Biological Activity

    DS96432529 (DS 96432529) is a potent and orally active bone anabolic agent with EC200 value of 0.024 ug/mL.
    DS96432529 exhibited the best PK profile and high in vitro activity, showed the highest in vivo efficacy, showed significant synergistic effects when combined with alendronate or parathyroid hormone.
    The mechanism of action is most likely mediated through CDK8 inhibition.

    Physicochemical Properties

    M.Wt 378.491
    Formula C18H26N4O3S
    Appearance Solid
    CAS No.
    Storage
    Solide Powder
    -20°C 12 Months; 4°C 6 Months
    In Solvent
    -80°C 6 Months; -20°C 6 Months
    Shipping
    Solubility

    10 mM in DMSO
    Chemical Name/SMILES

    3-amino-4-{(3S)-3-[(2-ethoxyethoxy)methyl]piperidin-1-yl}thieno[2,3-b]pyridine-2-carboxamide

    References

    1. Keiji Saito, et al. Bioorg Med Chem Lett. 2021 Dec 15;54:128440.

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