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Dagrocorat

Chemical Structure : Dagrocorat

CAS No.: 1044535-52-5

Dagrocorat (PF-00251802, PF 00251802)

Catalog No.: PC-61850Not For Human Use, Lab Use Only.

Dagrocorat (PF 00251802) is a potent, selective high-affinity dissociated agonist of the glucocorticoid receptor..

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Purity & Documentation Purity: >98% (HPLC) Select Batch:

    Biological Activity

    Dagrocorat (PF 00251802) is a potent, selective high-affinity dissociated agonist of the glucocorticoid receptor.

    Physicochemical Properties

    M.Wt 494.558
    Formula C29H29F3N2O2
    Appearance Solid
    CAS No.
    Storage
    Solide Powder
    -20 °C 12 Months; 4°C 6 Months
    In Solvent
    -80 °C 6 Months; -20°C 6 Months
    Shipping
    Solubility

    10 mM in DMSO

    Chemical Name/SMILES

    (4bR,7S,8aR)-4b-benzyl-7-hydroxy-N-(2-methylpyridin-3-yl)-7-(trifluoromethyl)-4b,5,6,7,8,8a,9,10-octahydrophenanthrene-2-carboxamide

    References

    1. Ripp SL, et al. Clin Pharmacol Drug Dev. 2017 Nov 7. doi: 10.1002/cpdd.411.

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