ENT1-IN-39 | ENT1 inhibitor | Probechem Biochemicals

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Chemical Structure : ENT1-IN-39

ENT1-IN-39 (ENT-1 inhibitor 39)

Catalog No.: PC-60154Not For Human Use, Lab Use Only.

ENT1-IN-39 (ENT-1 inhibitor 39) is a potent adenosine transport activity of equilibrative nucleoside transporter I protein (ENT1) with IC50 of 26.9 nM.

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Biological Activity

ENT1-IN-39 (ENT-1 inhibitor 39) is a potent adenosine transport activity of equilibrative nucleoside transporter I protein (ENT1) with IC50 of 26.9 nM.
ENT1-IN-39 displays ENT1 inhibition and efficacy in L-687414-induced hyperlocomotion mouse model (99.5 inhibition at 30 mg/kg, i.p.)

Physicochemical Properties

M.Wt	427.508
Formula	C25H25N5O2
Appearance	Solid
CAS No.
Storage	Solide Powder -20 °C 12 Months; 4°C 6 Months	In Solvent -80 °C 6 Months; -20°C 6 Months
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Solubility	10 mM in DMSO
Chemical Name/SMILES	6-(3,3-dimethyl-6-(2-methylpyrimidin-5-yl)-2-oxoindolin-1-yl)-1,3,3-trimethyl-1,3-dihydro-2H-pyrrolo[2,3-b]pyridin-2-one

References

1. Gerard Rosse. ACS Med. Chem. Lett., 2017, 8 (10), pp 995-996.

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ENT1-IN-39 (ENT-1 inhibitor 39)

Biological Activity

Physicochemical Properties

References

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