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ENT1-IN-39

Chemical Structure : ENT1-IN-39

CAS No.: 2097508-70-6

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ENT1-IN-39 (ENT-1 inhibitor 39)

Catalog No.: PC-60154Not For Human Use, Lab Use Only.

ENT1-IN-39 (ENT-1 inhibitor 39) is a potent adenosine transport activity of equilibrative nucleoside transporter I protein (ENT1) with IC50 of 26.9 nM.

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Purity & Documentation Purity: >98% (HPLC) Select Batch:

    Biological Activity

    ENT1-IN-39 (ENT-1 inhibitor 39) is a potent adenosine transport activity of equilibrative nucleoside transporter I protein (ENT1) with IC50 of 26.9 nM.
    ENT1-IN-39 displays ENT1 inhibition and efficacy in L-687414-induced hyperlocomotion mouse model (99.5 inhibition at 30 mg/kg, i.p.)

    Physicochemical Properties

    M.Wt 427.508
    Formula C25H25N5O2
    Appearance Solid
    CAS No.
    Storage
    Solide Powder
    -20 °C 12 Months; 4°C 6 Months
    In Solvent
    -80 °C 6 Months; -20°C 6 Months
    Shipping
    Solubility

    10 mM in DMSO
    Chemical Name/SMILES

    6-(3,3-dimethyl-6-(2-methylpyrimidin-5-yl)-2-oxoindolin-1-yl)-1,3,3-trimethyl-1,3-dihydro-2H-pyrrolo[2,3-b]pyridin-2-one

    References

    1. Gerard Rosse. ACS Med. Chem. Lett., 2017, 8 (10), pp 995-996.

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