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ENX-101

Chemical Structure : ENX-101

CAS No.: 1213669-91-0

ENX-101 (ENX101)

Catalog No.: PC-24258Not For Human Use, Lab Use Only.

ENX-101 is a α2,α3,α5-selective γ-aminobutyric acid type A (GABAA) receptor partial positive allosteric modulator (PAM), deuterated analog of L-838,417.

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Purity & Documentation Purity: >98% (HPLC) Select Batch:

Biological Activity

ENX-101 is a α2,α3,α5-selective γ-aminobutyric acid type A (GABAA) receptor partial positive allosteric modulator (PAM), deuterated analog of L-838,417.

Physicochemical Properties

M.Wt 408.46
Formula C19H10D9F2N7O
Appearance Solid
CAS No.
Storage
Solide Powder
-20°C 12 Months; 4°C 6 Months
In Solvent
-80°C 6 Months; -20°C 6 Months
Shipping
Solubility

10 mM in DMSO

Chemical Name/SMILES

3-(2,5-difluorophenyl)-6-((1-methyl-1H-1,2,4-triazol-5-yl)methoxy)-7-(2-(methyl-d3)propan-2-yl-1,1,1,3,3,3-d6)-[1,2,4]triazolo[4,3-b]pyridazine

References

1. Serrats J, et al. Epilepsia. 2025 Mar 15. doi: 10.1111/epi.18340.

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