Chemical Structure : EPZ-011989 trifluoroacetate
CAS No.:
1598383-41-5
EPZ-011989 trifluoroacetate
(EPZ011989 trifluoroacetate)
Catalog No. : PC-45115Not For Human Use, Lab Use Only.
EPZ-011989 trifluoroacetate is a potent, selective, orally bioavailable inhibitor of EZH2 with Ki of < 3 nM.
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Purity & Documentation Purity:
>98% (HPLC) Select Batch: PC-4511501
Biological Activity
EPZ-011989 trifluoroacetate is a potent, selective, orally bioavailable inhibitor of EZH2 with Ki of < 3 nM.
Physicochemical Properties
M.Wt
719.8339
Formula
C37H52F3N5O6
Appearance
Solid
CAS No.
Storage
Solide Powder
-20 °C 12 Months; 4°C 6 Months
In Solvent
-80 °C 6 Months; -20°C 6 Months
Shipping
Solubility
DMSO: ≥ 34 mg/mL
Chemical Name/SMILES
Benzamide, N-[(1,2-dihydro-4,6-dimethyl-2-oxo-3-pyridinyl)methyl]-3-[ethyl[trans-4-[(2-methoxyethyl)methylamino]cyclohexyl]amino]-2-methyl-5-[3-(4-morpholinyl)-1-propyn-1-yl]-, 2,2,2-trifluoroacetate (1:x)
References
1. Campbell JE, et al. ACS Med Chem Lett.
2. Gardner EE, et al. Cancer Cell.
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