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Chemical Structure : EPZ-030456
Catalog No.: PC-70107Not For Human Use, Lab Use Only.
EPZ-030456 (EPZ030456) is a potent, selective SMYD3 inhibitor with biochem IC50 of 4 nM.
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EPZ-030456 (EPZ030456) is a potent, selective SMYD3 inhibitor with biochem IC50 of 4 nM; displays noncompetitive inhibition with respect to SAM and MEKK2 with Ki of 1.2 and 1.1 nM, respectively; has cellular potency (IC50=48 nM) suitable to probe the in vitro biology of SMYD3 inhibition.
| M.Wt | 572.121 | |
| Formula | C28H34ClN5O4S | |
| Appearance | Solid | |
| Storage |
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| Solubility |
10 mM in DMSO |
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1. Mitchell LH, et al. ACS Med Chem Lett. 2015 Aug 27;7(2):134-8.
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