EPZ028862 | SMYD3 inhibitor | Probechem Biochemicals

Chemical Structure : EPZ028862

Catalog No.: PC-21039Not For Human Use, Lab Use Only.

EPZ028862 is a potent, selective inhibitor of SMYD3 with biochemical IC50 of 1.8 nM, and function of cellular methylation IC50 of 32 nM.

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Purity & Documentation Purity: >98% (HPLC)

Biological Activity

EPZ028862 is a potent, selective inhibitor of SMYD3 with biochemical IC50 of 1.8 nM, and function of cellular methylation IC50 of 32 nM.

M.Wt	422.54
Formula	C20H30N4O4S
Appearance	Solid
CAS No.
Storage	Solide Powder -20°C 12 Months; 4°C 6 Months	In Solvent -80°C 6 Months; -20°C 6 Months
Shipping
Solubility	10 mM in DMSO
Chemical Name/SMILES	O=C(C1=NOC(C2CC2)=C1)NC3CC(N4S(=O)([C@H]5CC[C@H](N)CC5)=O)CCC4C3

1. Michael J Thomenius, et al. PLoS One. 2018 Jun 1;13(6):e0197372.