Chemical Structure : EPZ031686
CAS No.:
2095161-11-6
EPZ031686
(EPZ-031686, EPZ 031686)
Catalog No. : PC-45608Not For Human Use, Lab Use Only.
EPZ031686 (EPZ 031686) is a potent, selective, small molecule SMYD3 inhibitor (Biochem IC50=3 nM, Cell IC50= 36 nM).
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Purity & Documentation Purity:
>98% (HPLC) Select Batch: PC-4560801
Biological Activity
EPZ031686 (EPZ 031686) is a potent, selective, small molecule SMYD3 inhibitor (Biochem IC50=3 nM, Cell IC50= 36 nM).
Physicochemical Properties
M.Wt
591.0858
Formula
C26H34ClF3N4O4S
Appearance
Solid
CAS No.
Storage
Solide Powder
-20 °C 12 Months; 4°C 6 Months
In Solvent
-80 °C 6 Months; -20°C 6 Months
Shipping
Solubility
DMSO: ≥ 5.9 mg/mL
Chemical Name/SMILES
1H-Indole-5-carboxamide, 6-chloro-2,3-dihydro-2-oxo-N-[(3-endo)-8-[[[1-(4,4,4-trifluorobutyl)-4-piperidinyl]methyl]sulfonyl]-8-azabicyclo[3.2.1]oct-3-yl]-
References
1. Mitchell LH, et al. ACS Med Chem Lett.
2. Rajajeyabalachandran G, et al. Expert Opin Ther Targets.
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