ESG-1-61

Chemical Structure : ESG-1-61

Catalog No.: PC-24332Not For Human Use, Lab Use Only.

ESG-1-61 is a potent, selective antagonist/inverse agonist of dopamine D3 receptor (D3R) with Ki of 0.73 nM, EC50 of 3.36 nM (Go activation) and4.36 nM (β-arrestin2 recruitment), show ~20-fold binding selectivity for D3 over D2 receptors.

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Biological Activity

Physicochemical Properties

M.Wt	466.06
Formula	C25H40ClN3O3
Appearance	Solid
CAS No.
Storage	Solide Powder -20°C 12 Months; 4°C 6 Months	In Solvent -80°C 6 Months; -20°C 6 Months
Shipping
Solubility	10 mM in DMSO
Chemical Name/SMILES	Propanamide, N-[trans-4-[2-[4-(3-chloro-5-ethyl-2-methoxyphenyl)-1-piperazinyl]ethyl]cyclohexyl]-3-methoxy-

References

1. Soler-Cedeño O, et al. Br J Pharmacol. 2025 Mar 27. doi: 10.1111/bph.70021.

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ESG-1-61

Biological Activity

Physicochemical Properties

References

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