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Chemical Structure : Elagolix
CAS No.: 834153-87-6
Catalog No.: PC-23475Not For Human Use, Lab Use Only.
Elagolix (NBI-56418) is a highly effective, selective, orally bioavailable, non-peptide gonadotropin-releasing hormone receptor (GnRH) antagonist with KD value of 54 pM.
| Packing | Price | Stock | Quantity |
|---|---|---|---|
| 5 mg | $88 | In stock | |
| 10 mg | $128 | In stock | |
| 25 mg | $228 | In stock | |
| 50 mg | Get quote | ||
| 100 mg | Get quote |
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Elagolix (NBI-56418) is a highly effective, selective, orally bioavailable, non-peptide gonadotropin-releasing hormone receptor (GnRH) antagonist with KD value of 54 pM.
| M.Wt | 631.60 | |
| Formula | C32H30F5N3O5 | |
| Appearance | Solid | |
| Storage |
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| Solubility |
10 mM in DMSO |
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| Chemical Name/SMILES |
(R)-4-((2-(5-(2-Fluoro-3-methoxyphenyl)-3-(2-fluoro-6-(trifluoromethyl)benzyl)-4-methyl-2,6-dioxo-3,6-dihydropyrimidin-1(2H)-yl)-1-phenylethyl)amino)butanoic acid |
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1. Kim SM, et al. J Med Chem. 2016 Oct 13;59(19):9150-9172. Epub 2016 Sep 27.
2. Chen C, et al. J Med Chem. 2008 Dec 11;51(23):7478-85.
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