Cat. No. |
Product Name |
Information |
PC-20087 |
TAK-385
GnRH receptor inhibitor
|
TAK-385 (Relugolix, TAK385) is a potent, orally active, non-peptide antagonist of human gonadotropin-releasing hormone (GnRH) receptor, inhibits GnRH-stimulated AA release from CHO cells expressing human GnRH receptor with IC50 of 0.85 nM. |
PC-61385 |
Linzagolix
GnRH antagonist
|
Linzagolix (KLH-2109, OBE-2109) is a novel potent gonadotrophin releasing hormone (GnRH) antagonist. |
PC-20045 |
Merigolix
GnRH receptor inhibitor
|
Merigolix is a potent, selective gonadotrophin releasing hormone (GnRH) antagonist. |
PC-38730 |
BAY1214784
GnRH-R antagonist
|
BAY 1214784 (BAY-784) is an orally available, potent, and selective antagonist of gonadotropin-releasing hormone receptor (GnRH-R) with IC50 of 21/ 24/ 35 nM for human/rat/cynomolgus GnRH-R, respectively. |
PC-38090 |
GnRH antagonist 2
|
GnRH antagonist 2 is a GnRH receptor antagonist that can be used for endometriosis research.. |
PC-43103 |
Leuprorelin
|
Leuprorelin (Leuprolide) is a GnRH analog and agonist of GnRH receptor, interrupts the normal pulsatile stimulation and desensitizing of the GnRH receptors.. |
PC-43101 |
Triptorelin
|
Triptorelin is a synthetic decapeptide agonist analog of luteinizing hormone releasing hormone (LHRH), shows greater potency than endogenous LHRH, triptorelin reversibly represses gonadotropin secretion.. |
PC-61391 |
Opigolix
|
A novel potent gonadotrophin releasing hormone (GnRH) antagonist.. |