Welcome to ProbeChem!Global Supplier of Chemical Probes, Inhibitors & Agonists.
EN | CN

You are here:Home-Chemical Inhibitors & Agonists-GPCR-P2Y Receptor-Elinogrel
Elinogrel

Chemical Structure : Elinogrel

CAS No.: 936500-94-6

Elinogrel (PRT-060128, PRT060128)

Catalog No.: PC-61587Not For Human Use, Lab Use Only.

Elinogrel (PRT060128) is a selective, reversible, competitive and direct-acting P2Y12 receptor antagonist with IC50 of 20 nM.

Packing Price Stock Quantity
5 mg $118 In stock
10 mg $188 In stock
25 mg $298 In stock
50 mg $498 In stock
100 mg Get quote

Bulk size, bulk discount!

E-mail: sales@probechem.com

Tech Support: tech@probechem.com

Purity & Documentation Purity: >98% (HPLC) Select Batch:

Biological Activity

Elinogrel (PRT060128) is a selective, reversible, competitive and direct-acting P2Y12 receptor antagonist with IC50 of 20 nM.
Elinogrel (PRT060128) shows potent antiplatelet effects for the treatment of acute coronary syndrome and prevention of secondary thrombotic events.

Physicochemical Properties

M.Wt 523.945
Formula C20H15ClFN5O5S2
Appearance Solid
CAS No.
Storage
Solide Powder
-20 °C 12 Months; 4°C 6 Months
In Solvent
-80 °C 6 Months; -20°C 6 Months
Shipping
Solubility

10 mM in DMSO

Chemical Name/SMILES

N-[4-(6-Fluoro-7-methylamino-2,4-dioxo-1,4-dihydro-2H-quinazolin-3-yl)phenyl]-N'-[(5-chlorothiophen-2-yl)sulfonyl]urea

References

1. Siller-Matula JM, et al. Br J Pharmacol. 2010 Feb 1;159(3):502-17.

2. Leonardi S, et al. Am Heart J. 2010 Jul;160(1):65-72.

3. Oestreich JH. Curr Opin Investig Drugs. 2010 Mar;11(3):340-8.

4. André P, et al. J Pharmacol Exp Ther. 2011 Jul;338(1):22-30.

Copyright © 2022 probechem.com. All Rights Reserved. probechem Copyright

Contact Us sales@probechem.com

Bulk Inquiry

* Indicates a Required FieldYour information is safe with us.

  • *Product name:
  • *Applicant name:
  • *Email address:
  • *Organization name:
  • *Requested quantity:
  • *Country:
  • *Additional Information:

Get Quote

* Indicates a Required FieldYour information is safe with us.

  • *Product name:
  • *Applicant name:
  • *Email address:
  • *Organization name:
  • *Requested quantity:
  • *Country:
  • Additional Information: