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Elobixibat

Chemical Structure : Elobixibat

CAS No.: 439087-18-0

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Elobixibat (A3309, AZD7806, AJG-533)

Catalog No.: PC-61407Not For Human Use, Lab Use Only.

Elobixibat (A3309, AZD7806, AJG-533) is an orally available, potent and selective apical sodium-dependent bile acid transporter (ASBT, ileal bile acid transporter (IBAT) and SLC10A2) inhibitor with IC50 of 0.53 nM, 0.13 nM, and 5.8 nM for human, mouse, and canine IBAT respectively.

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25 mg $598 In stock
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Purity & Documentation Purity: >98% (HPLC) Select Batch:

Biological Activity

Elobixibat (A3309, AZD7806, AJG-533) is an orally available, potent and selective apical sodium-dependent bile acid transporter (ASBT, ileal bile acid transporter (IBAT) and SLC10A2) inhibitor with IC50 of 0.53 nM, 0.13 nM, and 5.8 nM for human, mouse, and canine IBAT respectively.

Physicochemical Properties

M.Wt 695.89
Formula C36H45N3O7S2
Appearance Solid
CAS No.
Storage
Solide Powder
-20 °C 12 Months; 4°C 6 Months
In Solvent
-80 °C 6 Months; -20°C 6 Months
Shipping
Solubility

10 mM in DMSO
Chemical Name/SMILES

Glycine, (2R)-N-[[[3,3-dibutyl-2,3,4,5-tetrahydro-7-(methylthio)-1,1-dioxido-5-phenyl-1,5-benzothiazepin-8-yl]oxy]acetyl]-2-phenylglycyl- (9CI)

References

1. Chey WD, et al. Gastroenterol. 2014 May;109(5):782.

2. Wong BS, et al. Expert Opin Investig Drugs. 2013 Feb;22(2):277-84.

3. Wong BS, et al. Am J Gastroenterol. 2011 Dec;106(12):2154-64.

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