Equilin | 3βHSD1 inhibitor | Probechem Biochemicals

Chemical Structure : Equilin

CAS No.: 474-86-2

Equilin (7-Dehydroestrone)

Catalog No.: PC-21635Not For Human Use, Lab Use Only.

Equilin (7-Dehydroestrone) is a highly potent 3βHSD1 inhibitor with IC50 of 2.8 nM in VCaP cells, also inhibits the activity of purified 3βHSD1 with SPR KD of 2.23 uM.

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Biological Activity

Equilin (7-Dehydroestrone) is a highly potent 3βHSD1 inhibitor with IC50 of 2.8 nM in VCaP cells, also inhibits the activity of purified 3βHSD1 with SPR KD of 2.23 uM.
Equilin has a higher affinity to 3βHSD1 than BCA.
Equilin suppresses UBE3D-related tumor aggressiveness.

Physicochemical Properties

M.Wt	268.36
Formula	C18H20O2
Appearance	Solid
CAS No.
Storage	Solide Powder -20°C 12 Months; 4°C 6 Months	In Solvent -80°C 6 Months; -20°C 6 Months
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Solubility	10 mM in DMSO
Chemical Name/SMILES	(9S,13S,14S)-3-Hydroxy-13-methyl-6,9,11,12,13,14,15,16-octahydro-17H-cyclopenta[a]phenanthren-17-one

References

1. Xuebin Zhang, et al. J Clin Invest. 2023 Dec 15;133(24):e171199.

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Equilin (7-Dehydroestrone)

Biological Activity

Physicochemical Properties

References

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