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Chemical Structure : Equilin
CAS No.: 474-86-2
Catalog No.: PC-21635Not For Human Use, Lab Use Only.
Equilin (7-Dehydroestrone) is a highly potent 3βHSD1 inhibitor with IC50 of 2.8 nM in VCaP cells, also inhibits the activity of purified 3βHSD1 with SPR KD of 2.23 uM.
| Packing | Price | Stock | Quantity |
|---|---|---|---|
| 5 mg | $158 | In stock | |
| 10 mg | $248 | In stock | |
| 25 mg | $398 | In stock | |
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| 100 mg | Get quote |
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Equilin (7-Dehydroestrone) is a highly potent 3βHSD1 inhibitor with IC50 of 2.8 nM in VCaP cells, also inhibits the activity of purified 3βHSD1 with SPR KD of 2.23 uM.
Equilin has a higher affinity to 3βHSD1 than BCA.
Equilin suppresses UBE3D-related tumor aggressiveness.
| M.Wt | 268.36 | |
| Formula | C18H20O2 | |
| Appearance | Solid | |
| Storage |
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| Solubility |
10 mM in DMSO |
|
| Chemical Name/SMILES |
(9S,13S,14S)-3-Hydroxy-13-methyl-6,9,11,12,13,14,15,16-octahydro-17H-cyclopenta[a]phenanthren-17-one |
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1. Xuebin Zhang, et al. J Clin Invest. 2023 Dec 15;133(24):e171199.
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