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FAUC 1104

Chemical Structure : FAUC 1104

CAS No.: 1869983-86-7

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FAUC 1104 (FAUC1104, FAUC-1104)

Catalog No.: PC-61171Not For Human Use, Lab Use Only.

FAUC 1104 is a potent, biased allosteric agonist of CXCR3 (pEC50=5.22) that activates solely G proteins, induces chemotaxis, but fails to induce receptor internalization or β-arrestin 2 recruitment.

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Purity & Documentation Purity: >98% (HPLC) Select Batch:

    Biological Activity

    FAUC 1104 is a potent, biased allosteric agonist of CXCR3 (pEC50=5.22) that activates solely G proteins, induces chemotaxis, but fails to induce receptor internalization or β-arrestin 2 recruitment.

    Physicochemical Properties

    M.Wt 774.959
    Formula C46H54N4O7
    Appearance Solid
    CAS No.
    Storage
    Solide Powder
    -20 °C 12 Months; 4°C 6 Months
    In Solvent
    -80 °C 6 Months; -20°C 6 Months
    Shipping
    Solubility

    10 mM in DMSO
    Chemical Name/SMILES

    tert-Butyl {(S)-1-[(2,2-diphenylethyl)amino]-6-[(S)-2-(4-(4-methoxyphenyl)-4-oxobutanoyl)-1,2,3,4-tetrahydroisoquinoline-3-carboxamido]-1-oxohexan-2-yl}carbamate

    References

    1. Milanos L, et al. J Med Chem. 2016 Mar 10;59(5):2222-43.

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