Feniralstat (KVD-824) | Kallikrein inhibitor

Chemical Structure : Feniralstat

Feniralstat (KVD-824, KVD824)

Catalog No.: PC-73418Not For Human Use, Lab Use Only.

Feniralstat (KVD-824) is a potent, selective kallikrein inhibitor with IC50 of 6.7 nM for human plasma kallikrein (pKal), dispays no inhibition against human KLKl, FXIa and Factor Xlla (IC50>40 uM).

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Biological Activity

Feniralstat (KVD-824) is a potent, selective kallikrein inhibitor with IC50 of 6.7 nM for human plasma kallikrein (pKal), dispays no inhibition against human KLKl, FXIa and Factor Xlla (IC50>40 uM).

Physicochemical Properties

M.Wt	509.514
Formula	C26H25F2N5O4
Appearance	Solid
CAS No.
Storage	Solide Powder -20°C 12 Months; 4°C 6 Months	In Solvent -80°C 6 Months; -20°C 6 Months
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Solubility	10 mM in DMSO
Chemical Name/SMILES	1-(4-((5-fluoro-2-oxopyridin-1(2H)-yl)methyl)benzyl)-N-((3-fluoro-4-methoxypyridin-2-yl)methyl)-3-(methoxymethyl)-1H-pyrazole-4-carboxamide

References

1. Rebecca Louise DAVIE, et al. Pyrazole derivatives as plasma kallikrein inhibitors. WO2017207983A1. (Compound 30).

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Feniralstat (KVD-824, KVD824)

Biological Activity

Physicochemical Properties

References

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