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Filapixant

Chemical Structure : Filapixant

CAS No.: 1948232-63-0

Filapixant (BAY1902607, BAY 1902607)

Catalog No.: PC-20738Not For Human Use, Lab Use Only.

Filapixant (BAY1902607) is a potent, selective P2X3 receptor antagonist, shows a substantially higher in vitro selectivity for P2X3 over P2X2 when compared with Eliapixant (BAY1817080, Cat# PC-72754).

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Purity & Documentation Purity: >98% (HPLC) Select Batch:

Biological Activity

Filapixant (BAY1902607) is a potent, selective P2X3 receptor antagonist, shows a substantially higher in vitro selectivity for P2X3 over P2X2 when compared with Eliapixant (BAY1817080, Cat# PC-72754).
Filapixant has a higher in vitro selectivity for P2X3 than other receptor antagonists such as gefapixant, or even eliapixant.

Physicochemical Properties

M.Wt 521.56
Formula C24H26F3N5O3S
Appearance Solid
CAS No.
Storage
Solide Powder
-20°C 12 Months; 4°C 6 Months
In Solvent
-80°C 6 Months; -20°C 6 Months
Shipping
Solubility

10 mM in DMSO

Chemical Name/SMILES

3-(((R)-4-methylmorpholin-2-yl)methoxy)-5-(5-methylthiazol-2-yl)-N-((R)-1-(2-(trifluoromethyl)pyrimidin-5-yl)ethyl)benzamide

References

1. Davenport AJ, et, al. 1,3-thiazol-2-yl substituted benzamides. WO2016091776A1.

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