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Chemical Structure : GAT100
Catalog No.: PC-35488Not For Human Use, Lab Use Only.
GAT-100 (GAT100) is a potent, selective CB1R negative allosteric modulator (NAM) with cAMP EC50 and β-arr EC50 of 174 nM and 2.1 nM, does not exhibit inverse agonism.
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GAT-100 (GAT100) is a potent, selective CB1R negative allosteric modulator (NAM) with cAMP EC50 and β-arr EC50 of 174 nM and 2.1 nM, does not exhibit inverse agonism.
GAT-100 is a covalent probe for mapping structure-function correlates characteristic of the druggable CB1R allosteric space.
| M.Wt | 432.59 | |
| Formula | C25H28N4OS | |
| Appearance | Solid | |
| Storage |
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| Solubility |
10 mM in DMSO |
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1. Kulkarni PM, et al. J Med Chem. 2016 Jan 14;59(1):44-60.
2. Laprairie RB, et al. ACS Chem Neurosci. 2016 Jun 15;7(6):776-98.
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